Tailored Aza‐Michael Addition as Key Step in the Synthesis of 1 <i>H</i> ‐imidazo[5,1‐ <i>c</i> ][1,4]oxazine Scaffolds
نویسندگان
چکیده
A new strategy has been proposed for the synthesis of an array imidazo[5,1-c][1,4]oxazine chemotypes by using a planned aza-Michael addition in 3-CR heteroring-forming, post-cyclization transformation followed intramolecular fused-heterocycles formation process.
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ژورنال
عنوان ژورنال: European Journal of Organic Chemistry
سال: 2022
ISSN: ['1434-193X', '1099-0690']
DOI: https://doi.org/10.1002/ejoc.202201053